Structure-activity relationships and pharmacological profiles of new 5-HT, receptor agonists as antimigraine agents

  • Michel Ferez
  • , Gareth W. John

Research output: Contribution to journalArticlepeer-review

6 Scopus citations

Abstract

The design of new generation drugs acting as 5-HT, receptor agonists, in the field of acute treatment of migraine, is still very active. The reason is the need for safer medicines with improved response rates and a reduced rate of headache recurrence. This review focuses on the different classes of drugs, which have been classified based on the target upon which they act rather than upon structural cliaracterislics. Short SAR studies are reported for each series with a detailed pharmacological profile for the most interesting compounds. Keywords 5-HT, agonists, receptor selectivity, SAR

Original languageEnglish
Pages (from-to)304-310
Number of pages7
JournalCurrent Opinion in Drug Discovery and Development
Volume2
Issue number4
StatePublished - 1999
Externally publishedYes

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