(R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells

Dalia Barsyte-Lovejoy, Fengling Li, Menno J. Oudhoff, John H. Tatlock, Aiping Dong, Hong Zeng, Hong Wu, Spencer A. Freeman, Matthieu Schapira, Guillermo A. Senisterra, Ekaterina Kuznetsova, Richard Marcellus, Abdellah Allali-Hassani, Steven Kennedy, Jean Philippe Lambert, Amber L. Couzens, Ahmed Aman, Anne Claude Gingras, Rima Al-Awar, Paul V. FishBrian S. Gerstenberger, Lee Roberts, Caroline L. Benn, Rachel L. Grimley, Mitchell J.S. Braam, Fabio M.V. Rossi, Marius Sudol, Peter J. Brown, Mark E. Bunnage, Dafydd R. Owen, Colby Zaph, Masoud Vedadi, Cheryl H. Arrowsmith

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156 Scopus citations

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Biochemistry, Genetics and Molecular Biology